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1

Radiosynthesis of (E)-N-(2-[11C]methoxybenzyl)-3-phenyl-acrylamidine, a novel subnanomolar NR2B subtype-selective NMDA receptor antagonist

Cyrille Thominiaux, Béatrice de Bruin, Yann Bramoullé, Françoise Hinnen, Stéphane Demphel, Heric Valette, Michel Bottlaender, Laurent Besret, Michael Kassiou, Frédéric Dollé

Journal:

Applied Radiation and Isotopes

Year:

2006

Language:

english

File:

PDF, 198 KB

english, 2006

2

First Demonstration of Positive Allosteric-like Modulation at the Human Wild Type Translocator Protein (TSPO)

Narlawar, Rajeshwar, Werry, Eryn L., Scarf, Alana M., Hanani, Raphy, Chua, Sook Wern, King, Victoria A., Barron, Melissa L., Martins, Ralph N., Ittner, Lars M., Rendina, Louis M., Kassiou, Michael

Journal:

Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.84 MB

english, 2015

3

Translational evaluation of translocator protein as a marker of neuroinflammation in schizophrenia

Notter, T, Coughlin, J M, Gschwind, T, Weber-Stadlbauer, U, Wang, Y, Kassiou, M, Vernon, A C, Benke, D, Pomper, M G, Sawa, A, Meyer, U

Journal:

Molecular Psychiatry

Year:

2017

Language:

english

File:

PDF, 4.19 MB

english, 2017

4

The evolving science of phytocannabinoids

Reekie, Tristan A., Scott, Michael P., Kassiou, Michael

Journal:

Nature Reviews Chemistry

Year:

2017

Language:

english

File:

PDF, 1.76 MB

english, 2017

5

Preparation of a bromine-76 labelled analogue of epibatidine: a potent ligand for nicotinic acetylcholine receptor studies

M Kassiou, C Loc’h, F Dolle, J.L Musachio, L Dolci, C Crouzel, R.F Dannals, B Mazière

Journal:

Applied Radiation and Isotopes

Year:

2002

Language:

english

File:

PDF, 104 KB

english, 2002

6

Small animal SPECT and its place in the matrix of molecular imaging technologies

Meikle, Steven R, Kench, Peter, Kassiou, Michael, Banati, Richard B

Journal:

Physics in Medicine and Biology

Year:

2005

Language:

english

File:

PDF, 653 KB

english, 2005

7

The Nonpeptide Oxytocin Receptor Agonist WAY 267,464: Receptor-Binding Profile, Prosocial Effects and Distribution of c-Fos Expression in Adolescent Rats

C. Hicks, W. Jorgensen, C. Brown, J. Fardell, J. Koehbach, C. W. Gruber, M. Kassiou, G. E. Hunt, I. S. McGregor

Journal:

Journal of Neuroendocrinology

Year:

2012

Language:

english

File:

PDF, 1.03 MB

english, 2012

8

Boron in Drug Discovery: Carboranes as Unique Pharmacophores in Biologically Active Compounds

Issa, Fatiah, Kassiou, Michael, Rendina, Louis M.

Journal:

Chemical Reviews

Year:

2011

Language:

english

File:

PDF, 5.27 MB

english, 2011

9

The translocator protein (TSPO): A novel target for cancer chemotherapy

Austin, Christopher J.D., Kahlert, Jan, Kassiou, Michael, Rendina, Louis M.

Journal:

The International Journal of Biochemistry & Cell Biology

Year:

2013

Language:

english

File:

PDF, 978 KB

english, 2013

10

A practical synthesis of (1S,4S)-2,5-diazabicyclo[2.2.1]heptane

Beinat, Corinne, Banister, Samuel D., McErlean, Christopher S.P., Kassiou, Michael

Journal:

Tetrahedron Letters

Year:

2013

Language:

english

File:

PDF, 544 KB

english, 2013

11

Improved accessibility to the desoxy analogues of Δ9-tetrahydrocannabinol and cannabidiol

Wilkinson, Shane M., Price, Jason, Kassiou, Michael

Journal:

Tetrahedron Letters

Year:

2013

Language:

english

File:

PDF, 573 KB

english, 2013

12

The Translocator Protein

Scarf, A. M., Kassiou, M.

Journal:

Journal of Nuclear Medicine

Year:

2011

Language:

english

File:

PDF, 930 KB

english, 2011

13

Is there Any Correlation Between Binding and Functional Effects at the Translocator Protein (TSPO) (18 kDa)?

M. Scarf, A., M. Auman, K., Kassiou, M.

Journal:

Current Molecular Medicine

Year:

2012

Language:

english

File:

PDF, 868 KB

english, 2012

14

Development of Radioligands for In Vivo Imaging of GABAA-Benzodiazepine Receptors

Katsifis, Andrew, Kassiou, Michael

Journal:

Mini Reviews in Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 259 KB

english, 2004

15

Structural Optimization and Pharmacological Evaluation of Inhibitors Targeting Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases (DYRK) and CDC-like kinases (CLK) in Glioblastoma

Zhou, Qingqing, Phoa, Athena F., Abbassi, Ramzi H., Hoque, Monira, Reekie, Tristan A., Font, Josep S., Ryan, Renae M., Stringer, Brett W., Day, Bryan W., Johns, Terrance G., Munoz, Lenka, Kassiou, Mic

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.29 MB

english, 2017

16

Cubanes in Medicinal Chemistry

Reekie, Tristan, Williams, Craig Mckenzie, Rendina, Louis M, Kassiou, Michael

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.17 MB

english, 2018

17

Targeting the Oxytocin System: New Pharmacotherapeutic Approaches

Gulliver, Damien, Werry, Eryn, Reekie, Tristan A., Katte, Timothy A., Jorgensen, William, Kassiou, Michael

Journal:

Trends in Pharmacological Sciences

Year:

2018

Language:

english

File:

PDF, 3.28 MB

english, 2018

18

Synthesis and in vitro evaluation of fluorine-18 benzimidazole sulfones as CB2 PET-radioligands

Kallinen, Annukka, Boyd, Rochelle, Lane, Samuel, Bhalla, Rajiv, Mardon, Karine, Stimson, Damion H. R., Werry, Eryn L., Fulton, Roger, Connor, Mark, Kassiou, Michael

Journal:

Organic & Biomolecular Chemistry

Year:

2019

Language:

english

File:

PDF, 3.89 MB

english, 2019

19

Imaging disease activity of rheumatoid arthritis by macrophage targeting using second generation translocator protein positron emission tomography tracers

Bruijnen, S. T. G., Verweij, N. J. F., Gent, Y. Y. J., Huisman, M. C., Windhorst, A. D., Kassiou, M., van de Ven, P. M., Lammertsma, A. A., Hoekstra, O. S., Voskuyl, A. E., van der Laken, C. J., Wolos

Journal:

Year:

2019

Language:

english

File:

PDF, 909 KB

english, 2019

20

Letter: Myocardial infarction on a 17-year-old diabetic adolescent

Bartsocas, C.S., Kassiou, C., Dafogianni, C.

Journal:

Diabetic Medicine

Year:

1998

Language:

english

File:

PDF, 19 KB

english, 1998

21

Synthesis of iodine-123 labelled analogues of the partial agonist (S)- and (R)-bretazenil for the study of CNS benzodiazepine receptors using SPECT

Andrew Katsifis, Filomena Mattner, Meredith McPhee, Michael Kassiou, Ljubco Najdovski, Branko Dikic

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1996

Language:

english

File:

PDF, 673 KB

english, 1996

22

Synthesis of iodine-123 labelled analogues of imidazenil and ethyl-imidazenil for studying benzodiazepine receptors using SPECT

Andrew Katsifis, Filomena Mattner, Branko Dikic, Ljubco Najdovski, Michael Kassiou

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1996

Language:

english

File:

PDF, 608 KB

english, 1996

23

Synthesis of 3-[(1-[11C]methyl-2(S)-pyrrolidinyl) methoxy]pyridine and 3-[(1-[11C]methyl-2(R)-pyrrolidinyl) methoxy]pyridine: Radioligands for in vivo studies of neuronal nicotinic acetylcholine receptors

Michael Kassiou, Hayden T. Ravert, William B. Mathews, John L. Musachio, Edythe D. London, Robert F. Dannals

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1997

File:

PDF, 443 KB

1997

24

Radiosynthesis of bromine-76 and iodine-123 labelled enantiomers of A-69024: radioligands for dopamine D1 receptor studies using PET and SPECT

Michael Kassiou, Christian Loc'h, Andrew Katsifis, Vahan Papazian, Filomena Mattner, Branko Dikic, Bernard Mazière

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2000

File:

PDF, 260 KB

2000

25

ChemInform Abstract: Synthesis and Evaluation of Halogenated Dibenzodiazepines as Muscarinic Receptor Ligands.

M. KASSIOU, R. W. READ, X. SHI

Journal:

Year:

1997

File:

PDF, 30 KB

1997

26

ChemInform Abstract: Recent Advances in the Mitsunobu Reaction. Modifications and Applications to Biologically Active Molecules

A. J. Reynolds, M. Kassiou

Journal:

Year:

2010

File:

PDF, 24 KB

2010

27

Radiosynthesis of [18F]DPA-714, a selective radioligand for imaging the translocator protein (18 kDa) with PET

Annelaure Damont, Françoise Hinnen, Bertrand Kuhnast, Marie-Anne Schöllhorn-Peyronneau, Michelle James, Christopher Luus, Bertrand Tavitian, Michael Kassiou, Frédéric Dollé

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2008

Language:

english

File:

PDF, 193 KB

english, 2008

28

The development of PET radioligands for imaging the translocator protein (18 kDa): What have we learned?

Christopher Luus, Raphy Hanani, Aaron Reynolds, Michael Kassiou

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2010

Language:

english

File:

PDF, 208 KB

english, 2010

29

Radiosynthesis of (±)-1-(2-bromo-4,5-dimethoxybenzyl)-7-hydroxy-6-methoxy-2-[11C]-methyI-l,2,3,4-tetrahydro-isoquinoline, [11C]A-69024: A non-benzazepine antagonist for studying dopamine D1 receptors In vivo using PET

Michael Kassiou, William B. Mathews, John L. Musachio, Hayden T. Ravert, Richard M. Lambrecht, Robert F. Dannals

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1994

Language:

english

File:

PDF, 357 KB

english, 1994

30

Synthesis of [76Br]4-bromodexetimide and [76Br]4-bromolevetimide: Radiotracers for studying muscarinic cholinergic receptors using PET

Michael Kassiou, Christian Loc'h, Veronique Strijckmans, Andrew Katsifis, Richard M. Lambrecht, Mariannick Maziere, Bernard Maziere

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1995

Language:

english

File:

PDF, 359 KB

english, 1995

31

Radiosynthesis and in vivo evaluation of [11C]Ro-647312: a novel NR1/2B subtype selective NMDA receptor radioligand

Frédéric Dollé, Héric Valette, Stéphane Demphel, Christine Coulon, Michelle Ottaviani, Michel Bottlaender, Michael Kassiou

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2004

Language:

english

File:

PDF, 193 KB

english, 2004

32

Dopamine D1 receptor imaging in the rodent and primate brain using the isoquinoline (+)-[11C]A-69024 and positron emission tomography

Laurent Besret, Frédéric Dollé, Anne-Sophie Hérard, Martine Guillermier, Stéphane Demphel, Françoise Hinnen, Christine Coulon, Michèle Ottaviani, Michel Bottlaender, Philippe Hantraye, Michael Kassiou

Journal:

Journal of Pharmaceutical Sciences

Year:

2008

Language:

english

File:

PDF, 267 KB

english, 2008

33

3-Pyridyl ethers as SPECT radioligands for imaging nicotinic acetylcholine receptors

D.J Henderson, S Eberl, S Thomson, A Smith, R.D Allan, M.J Fulham, R Loiacono, M Kassiou

Journal:

Applied Radiation and Isotopes

Year:

2004

Language:

english

File:

PDF, 237 KB

english, 2004

34

Synthesis, radiosynthesis and In vivo evaluation of 5-[3-(4-Benzylpiperidin-1-yl)prop-1-ynyl]-1,3-dihydrobenzoimidazol-2-[11C]one, as a potent NR1A/2B subtype selective NMDA PET radiotracer

Gaëlle Roger, Béatrice Lagnel, Laurent Besret, Yann Bramoullé, Christine Coulon, Michelle Ottaviani, Michael Kassiou, Michel Bottlaender, Héric Valette, Frédéric Dollé

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 285 KB

english, 2003

35

Radiosynthesis and pharmacological evaluation of [11C]EMD-95885: a high affinity ligand for NR2B-containing NMDA receptors

G Roger, F Dollé, B de Bruin, X Liu, L Besret, Y Bramoullé, C Coulon, M Ottaviani, M Bottlaender, H Valette, M Kassiou

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 368 KB

english, 2004

36

Synthesis and in vitro evaluation of new benzovesamicol analogues as potential imaging probes for the vesicular acetylcholine transporter

Yolanda Zea-Ponce, Sylvie Mavel, Thaer Assaad, Shane E. Kruse, Stanley M. Parsons, Patrick Emond, Sylvie Chalon, Nicolas Giboureau, Michael Kassiou, Denis Guilloteau

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 349 KB

english, 2005

37

Synthesis and in vivo evaluation of a new PET radioligand for studying sigma-2 receptors

Michael Kassiou, Robert F. Dannals, Xiang Liu, Dean F. Wong, Hayden T. Ravert, Ursula A. Scheffel

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 120 KB

english, 2005

38

Synthesis and in vivo evaluation of a novel peripheral benzodiazepine receptor PET radioligand

Michelle L. James, Roger R. Fulton, David J. Henderson, Stefan Eberl, Steven R. Meikle, Sally Thomson, Robin D. Allan, Frederic Dolle, Michael J. Fulham, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 251 KB

english, 2005

39

Cubyl amides: Novel P2X7 receptor antagonists

Hendra Gunosewoyo, Jun Liu Guo, Maxwell R. Bennett, Mark J. Coster, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 268 KB

english, 2008

40

Positron Emission Tomography Imaging of Neuroinflammation

Annachiara Cagnin, Michael Kassiou, Steve R. Meikle, Richard B. Banati

Journal:

Neurotherapeutics

Year:

2007

Language:

english

File:

PDF, 235 KB

english, 2007

41

Trishomocubanes, a new class of selective and high affinity ligands for the sigma binding site

Michael Kassiou, Vu H. Nguyen, Robert Knott, MacDonald J. Christie, Trevor W. Hambley

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 279 KB

english, 1996

42

Improved synthesis of the peripheral benzodiazepine receptor ligand [11C]DPA-713 using [11C]methyl triflate

C. Thominiaux, F. Dollé, M.L. James, Y. Bramoullé, H. Boutin, L. Besret, M.-C. Grégoire, H. Valette, M. Bottlaender, B. Tavitian, Ph. Hantraye, S. Selleri, M. Kassiou

Journal:

Applied Radiation and Isotopes

Year:

2006

Language:

english

File:

PDF, 127 KB

english, 2006

43

Purinergic P2X7 receptor antagonists: Chemistry and fundamentals of biological screening

Hendra Gunosewoyo, Mark J. Coster, Maxwell R. Bennett, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 412 KB

english, 2009

44

Synthesis and in vitro evaluation of novel derivatives of diphenylsulfide as serotonin transporter ligands

Johnny Vercouillie, Sylvie Mavel, Laurent Galineau, Tiziana Ragusa, Robert Innis, Michael Kassiou, Sylvie Chalon, Frédéric Dollé, Jean-Claude Besnard, Denis Guilloteau, Patrick Emond

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 121 KB

english, 2006

45

Synthesis and in vitro evaluation of N-substituted aza-trozamicol analogs as vesicular acetylcholine transporter ligands

Thaer Assaad, Sylvie Mavel, Stanley M. Parsons, Shane Kruse, Laurent Galineau, Hassan Allouchi, Michael Kassiou, Sylvie Chalon, Denis Guilloteau, Patrick Emond

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 125 KB

english, 2006

46

Oxo-bridged isomers of aza-trishomocubane sigma (σ) receptor ligands: Synthesis, in vitro binding, and molecular modeling

Samuel D. Banister, Iman A. Moussa, Meredith J.T. Jordan, Mark J. Coster, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 492 KB

english, 2010

47

Pyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO)

Aaron Reynolds, Raphy Hanani, David Hibbs, Annelaure Damont, Eleonora Da Pozzo, Silvia Selleri, Frédéric Dollé, Claudia Martini, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 373 KB

english, 2010

48

Trishomocubane as a scaffold for the development of selective dopamine transporter (DAT) ligands

Samuel D. Banister, Iman A. Moussa, Corinne Beinat, Aaron J. Reynolds, Paolo Schiavini, William T. Jorgensen, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 309 KB

english, 2011

49

Molecular hybridization of 4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecane-3-ol with sigma (σ) receptor ligands modulates off-target activity and subtype selectivity

Samuel D. Banister, Iman A. Moussa, William T. Jorgensen, Sook Wern Chua, Michael Kassiou

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 408 KB

english, 2011

50

Water-soluble phosphonium salts containing 1,12-dicarba-closo-dodecaborane(12)

Joseph A. Ioppolo, Michael Kassiou, Louis M. Rendina

Journal:

Tetrahedron Letters

Year:

2009

Language:

english

File:

PDF, 245 KB

english, 2009